Local Anesthetic Sodium Block
unseel.com · lidocaine  ·  NaV channel  ·  use-dependent  ·  action potential
Na⁺ current 100%
channel resting
drug outside
state
NaV channel & membrane Neutral base (B) — crosses
Cation (BH⁺) — pore blocker Action potential fires
Unseel.com · Local Anesthetic Mechanism: How Lidocaine Blocks the Voltage-Gated Sodium Channel